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Target
Mu-type opioid receptor
Ligand
BDBM50008891
Substrate
n/a
Meas. Tech.
ChEMBL_146259 (CHEMBL757483)
Ki
>10000±n/a nM
Citation
 Vecchietti, V; Giordani, A; Giardina, G; Colle, R; Clarke, GD (2S)-1-(arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective kappa opioid analgesics. J Med Chem 34:397-403 (1991) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50008891
Synonyms:
2-(4-Fluoro-phenyl)-1-(2-pyrrolidin-1-ylmethyl-piperidin-1-yl)-ethanone(HCl) | CHEMBL128796
Type:
Small organic molecule
Emp. Form.:
C18H25FN2O
Mol. Mass.:
304.4023
SMILES:
Fc1ccc(CC(=O)N2CCCCC2CN2CCCC2)cc1
Structure:
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