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Target
Adenosine receptor A1
Ligand
BDBM82021
Substrate
n/a
Meas. Tech.
ChEMBL_29452 (CHEMBL641037)
Ki
3300±n/a nM
Citation
 Peet, NP; Dickerson, GA; Abdallah, AH; Daly, JW; Ukena, D Benzo[1,2-c:5,4-c']dipyrazoles: non-xanthine adenosine antagonists. J Med Chem 31:2034-9 (1988) [PubMed]  Article 
Target
Name:
Adenosine receptor A1
Synonyms:
AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1
Type:
Protein
Mol. Mass.:
36704.13
Organism:
Rattus norvegicus (rat)
Description:
n/a
Residue:
326
Sequence:
MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGALVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVTQRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYMVYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALILFLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFLKIWNDHFRCQPKPPIDEDLPEEKAED
  
Inhibitor
Name:
BDBM82021
Synonyms:
1,3-Diethylxanthine | CAS_101420 | CHEMBL416013 | NSC_101420
Type:
Small organic molecule
Emp. Form.:
C9H12N4O2
Mol. Mass.:
208.2172
SMILES:
CCn1c2nc[nH]c2c(=O)n(CC)c1=O
Structure:
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