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TargetAdenosine receptor A1
LigandBDBM50023505
Substrate/Competitorn/a
Meas. Tech.ChEBML_28547
IC50 31±n/a nM
Citation Francis, JECash, WDPsychoyos, SGhai, GWenk, PFriedmann, RCAtkins, CWarren, VFurness, PHyun, JL Structure-activity profile of a series of novel triazoloquinazoline adenosine antagonists. J Med Chem31:1014-20 (1988) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Adenosine receptor A1
Name:Adenosine receptor
Synonyms:ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptors A1
Type:Protein
Mol. Mass.:36704.13
Organism:Rattus norvegicus (rat)
Description:n/a
Residue:326
Sequence:
MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50023505
NameBDBM50023505
Synonyms:2-Furan-2-yl-9-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-5-ylamine | CHEMBL267015
TypeSmall organic molecule
Emp. Form.C14H11N5O2
Mol. Mass.281.2694
SMILESCOc1ccc2nc(N)n3nc(nc3c2c1)-c1ccco1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a