Reaction Details Report a problem with these data
Target
Platelet-activating factor acetylhydrolase [136-227]
Ligand
BDBM50040459
Substrate
n/a
Meas. Tech.
ChEMBL_156342 (CHEMBL759985)
IC50
1400±n/a nM
Citation
 Beaton, HG; Bennion, C; Connolly, S; Cook, AR; Gensmantel, NP; Hallam, C; Hardy, K; Hitchin, B; Jackson, CG; Robinson, DH Discovery of new non-phospholipid inhibitors of the secretory phospholipases A2. J Med Chem 37:557-9 (1994) [PubMed]  Article 
Target
Name:
Platelet-activating factor acetylhydrolase [136-227]
Synonyms:
A0A5G2RFL7_PIG | Group VII phospholipase A2 | PLA2G7
Type:
PROTEIN
Mol. Mass.:
10360.56
Organism:
Sus scrofa
Description:
ChEMBL_156342
Residue:
92
Sequence:
SPLRTGEKYPLIIFSHGLGAFRTIYSAIGTDLASYGFIVAAVEHRDGSASATYFFKDQSAAEIRNKTWLYLRTLGKGEEEFPLRNEQVRQRA
  
Inhibitor
Name:
BDBM50040459
Synonyms:
(R)-3-((S)-Decanoylamino)-5-methyl-hexanoic acid | CHEMBL152773
Type:
Small organic molecule
Emp. Form.:
C17H33NO3
Mol. Mass.:
299.4488
SMILES:
CCCCCCCCCC(=O)N[C@H](CC(C)C)CC(O)=O
Structure:
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