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Target
Mu-type opioid receptor
Ligand
BDBM50456334
Substrate
n/a
Meas. Tech.
ChEMBL_221917 (CHEMBL842482)
IC50
557±n/a nM
Citation
Yamazaki, T; Ro, S; Goodman, M; Chung, NN; Schiller, PW A topochemical approach to explain morphiceptin bioactivity. J Med Chem 36:708-19 (1993) [PubMed] Article
More Info.:
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI