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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50065136
Substrate/Competitorn/a
Meas. Tech.ChEMBL_200969
Ki 0.14±n/a nM
Citation John, CSLim, BBVilner, BJGeyer, BCBowen, WD Substituted halogenated arylsulfonamides: a new class of sigma receptor binding tumor imaging agents. J Med Chem41:2445-50 (1998) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Aging-associated gene 8 protein | SIG-1R | SR-BP | SR31747-binding protein | Sigma 1-type opioid receptor | Sigma opioid receptor | Sigma1R | hSigmaR1
Type:Enzyme Catalytic Domain
Mol. Mass.:25124.85
Organism:Homo sapiens (Human)
Description:Sigma 0 HUMAN::Q99720
Residue:223
Sequence:
MQWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLFGQDP
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  Blast E-value cutoff:
BDBM50065136
NameBDBM50065136
Synonyms:CHEMBL81455 | N-(2-Azepan-1-yl-ethyl)-4-iodo-N-methyl-benzenesulfonamide
TypeSmall organic molecule
Emp. Form.C15H23IN2O2S
Mol. Mass.422.325
SMILESCN(CCN1CCCCCC1)S(=O)(=O)c1ccc(I)cc1
Structure
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n/a