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Target
Lysophosphatidic acid receptor 1
Ligand
BDBM50177336
Substrate
n/a
Meas. Tech.
ChEMBL_329844 (CHEMBL862793)
Ki
497±n/a nM
Citation
 Gududuru, V; Zeng, K; Tsukahara, R; Makarova, N; Fujiwara, Y; Pigg, KR; Baker, DL; Tigyi, G; Miller, DD Identification of Darmstoff analogs as selective agonists and antagonists of lysophosphatidic acid receptors. Bioorg Med Chem Lett 16:451-6 (2005) [PubMed]  Article 
Target
Name:
Lysophosphatidic acid receptor 1
Synonyms:
Edg2 | Gpcr91 | LPAR1_RAT | Lpa1 | Lpar1 | Lysophosphatidic acid receptor 1/lysophosphatidic acid receptor 3 | Lysophosphatidic acid receptor Edg-2
Type:
PROTEIN
Mol. Mass.:
41130.42
Organism:
Rattus norvegicus
Description:
ChEMBL_329844
Residue:
364
Sequence:
MAAASTSSPVISQPQFTAMNEQQCFYNESIAFFYNRSGKYLATEWNTVSKLVMGLGITVCVFIMLANLLVMVAIYVNRRFHFPIYYLMANLAAADFFAGLAYFYLMFNTGPNTRRLTVSTWLLRQGLIDTSLTASVANLLAIAIERHITVFRMQLHTRMSNRRVVVVIVVIWTMAIVMGAIPSVGWNCICDIDHCSNMAPLYSDSYLVFWAIFNLVTFVVMVVLYAHIFGYVRQRTMRMSRHSSGPRRNRDTMMSLLKTVVIVLGAFIVCWTPGLVLLLLDVCCPQCDVLAYEKFFLLLAEFNSAMNPIIYSYRDKEMSATFRQILCCQRNENPNGPTEGSDRSASSLNHTILAGVHSNDHSVV
  
Inhibitor
Name:
BDBM50177336
Synonyms:
CHEMBL373007 | potassium (2-(heptadec-9-enyl)-1,3-dioxolan-4-yl)methyl hydrogenphosphate
Type:
Small organic molecule
Emp. Form.:
C21H40O6P
Mol. Mass.:
419.513
SMILES:
CCCCCCC\C=C\CCCCCCCCC1OCC(COP(O)([O-])=O)O1
Structure:
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