Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM29080
Substrate
n/a
Meas. Tech.
ChEMBL_342813 (CHEMBL868884)
Ki
>10000±n/a nM
Citation
 Appendino, G; Minassi, A; Berton, L; Moriello, AS; Cascio, MG; De Petrocellis, L; Di Marzo, V Oxyhomologues of anandamide and related endolipids: chemoselective synthesis and biological activity. J Med Chem 49:2333-8 (2006) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Homo sapiens (Human)
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM29080
Synonyms:
CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA | Oleoyl monoethanolamide | Oleoylethanolamide (OEA)
Type:
n/a
Emp. Form.:
C20H39NO2
Mol. Mass.:
325.5292
SMILES:
CCCCCCCC\C=C/CCCCCCCC(=O)NCCO
Structure:
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