| Reaction Details |
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 | Report a problem with these data |
| Target | Dopamine D5 receptor |
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| Ligand | BDBM50196234 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_417943 |
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| Ki | 0.61±n/a nM |
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| Citation |  Enzensperger, C; Lehmann, J Dopamine/serotonin receptor ligands. 13: Homologization of a benzindoloazecine-type dopamine receptor antagonist modulates the affinities for dopamine D(1)-D(5) receptors. J Med Chem49:6408-11 (2006) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Dopamine D5 receptor |
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| Name: | Dopamine receptor |
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| Synonyms: | D(1B) dopamine receptor | D(5) dopamine receptor | D1beta dopamine receptor | DOPAMINE D5 | DRD5 | Dopamine receptor | dopamine receptor D5 |
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| Type: | Protein |
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| Mol. Mass.: | 52943.41 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21918 |
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| Residue: | 477 |
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| Sequence: | MLPPGSNGTAYPGQFALYQQLAQGNAVGGSAGAPPLGPSQVVTACLLTLLIIWTLLGNVL
VCAAIVRSRHLRANMTNVFIVSLAVSDLFVALLVMPWKAVAEVAGYWPFGAFCDVWVAFD
IMCSTASILNLCVISVDRYWAISRPFRYKRKMTQRMALVMVGLAWTLSILISFIPVQLNW
HRDQAASWGGLDLPNNLANWTPWEEDFWEPDVNAENCDSSLNRTYAISSSLISFYIPVAI
MIVTYTRIYRIAQVQIRRISSLERAAEHAQSCRSSAACAPDTSLRASIKKETKVLKTLSV
IMGVFVCCWLPFFILNCMVPFCSGHPEGPPAGFPCVSETTFDVFVWFGWANSSLNPVIYA
FNADFQKVFAQLLGCSHFCSRTPVETVNISNELISYNQDIVFHKEIAAAYIHMMPNAVTP
GNREVDNDEEEGPFDRMFQIYQTSPDGDPVAESVWELDCEGEISLDKITPFTPNGFH
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| BDBM50196234 |
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| Name | BDBM50196234 |
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| Synonyms: | 8-methyl-5,6,7,8,9,10,15,16-octahydroindolo[3,2-g][4]benzazacycloundecine | CHEMBL216258 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H24N2 |
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| Mol. Mass. | 304.4287 |
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| SMILES | CN1CCCc2ccccc2Cc2[nH]c3ccccc3c2CC1 |
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| Structure | 
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| n/a |
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