Reaction Details Report a problem with these data
Target
Protein ADM2
Ligand
BDBM50246709
Substrate
n/a
Meas. Tech.
ChEMBL_556927 (CHEMBL954953)
IC50
418±n/a nM
Citation
Miranda, LP; Holder, JR; Shi, L; Bennett, B; Aral, J; Gegg, CV; Wright, M; Walker, K; Doellgast, G; Rogers, R; Li, H; Valladares, V; Salyers, K; Johnson, E; Wild, K Identification of potent, selective, and metabolically stable peptide antagonists to the calcitonin gene-related peptide (CGRP) receptor. J Med Chem 51:7889-97 (2008) [PubMed] Article
More Info.:
Target
Name:
Protein ADM2
Synonyms:
ADM2 | ADM2_HUMAN | AM2
Type:
PROTEIN
Mol. Mass.:
15883.28
Organism:
Homo sapiens (Human)
Description:
ChEMBL_556927
Residue:
148
Sequence:
MARIPTAALGCISLLCLQLPGSLSRSLGGDPRPVKPREPPARSPSSSLQPRHPAPRPVVWKLHRALQAQRGAGLAPVMGQPLRDGGRQHSGPRRHSGPRRTQAQLLRVGCVLGTCQVQNLSHRLWQLMGPAGRQDSAPVDPSSPHSYG