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Target
Glucose-6-phosphate 1-dehydrogenase
Ligand
BDBM50223368
Substrate
n/a
Meas. Tech.
ChEMBL_542429 (CHEMBL1010666)
Ki
1700±n/a nM
Citation
Cordeiro, AT; Thiemann, OH; Michels, PA Inhibition of Trypanosoma brucei glucose-6-phosphate dehydrogenase by human steroids and their effects on the viability of cultured parasites. Bioorg Med Chem 17:2483-9 (2009) [PubMed] Article
More Info.:
Target
Name:
Glucose-6-phosphate 1-dehydrogenase
Synonyms:
n/a
Type:
PROTEIN
Mol. Mass.:
59057.43
Organism:
Trypanosoma brucei
Description:
ChEMBL_542430
Residue:
521
Sequence:
MQNCRKVADTLRKDSCDIIPDAAAPELKERALTIVVLGASGDLARNKTFPALFQLFCNGLIPRTINIVGYARTKMPDVEQWKKESLAKHFPRAKDRCPHIEAFLKTITYISGSYDGADDFFRLNDVITKFEESFPGKQKGGNRLFYLALPPSVFMHACTGIRTHVMQKPGLGWVRIIIEKPFGHDTESSNELSRQLEPLFEESQIFRIDHYLGKEMVQNIVVTRFANRVFSALWNNNNIACVRITFKESIGTEGRGGYFDKAGIIRDVVQNHLTQILSLLAMEKPRSLSPEDIRDEKVIVLRHVNPVTPADCVLGQYTRSEDGSIPGYLEDPTVPRGSKCATFVVLRLFINNDRWDGVPFIIEAGKAVERRYLGIRIQFKDEIRPFGVAAQRNELIIRAQPSEAMYLRLTAKTPGVLSDTHQTELDLSYEHRYNITLPDAYESLIHEALLGRSTNFVRKDELDAAWRIYTPLLEAIERGETTTYPYSAGSKGPAEAQKFVDDTGFKPLTGDIYQQRKLHHL