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TargetMu-type opioid receptor
LigandBDBM50336661
Substrate/Competitorn/a
Meas. Tech.ChEMBL_722917
Ki 0.134±n/a nM
Citation Nemoto, TYamamoto, NWatanabe, AFujii, HHasebe, KNakajima, MMochizuki, HNagase, H Synthesis of 6,14-epoxymorphinan derivatives and their pharmacologies. Bioorg Med Chem19:1205-21 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50336661
NameBDBM50336661
Synonyms:CHEMBL1672475 | N-{[(1R,9R,10S,13S)-17-(cyclopropylmethyl)-4-hydroxy-18-oxa-17-azapentacyclo[7.5.3.1^{10,13}.0^{1,10}.0^{2,7}]octadeca-2(7),3,5-trien-13-yl]methyl}benzamide
TypeSmall organic molecule
Emp. Form.C28H32N2O3
Mol. Mass.444.5653
SMILESOc1ccc2C[C@H]3N(CC4CC4)CC[C@@]4(C[C@]5(CNC(=O)c6ccccc6)CC[C@@]34O5)c2c1 |r,THB:8:7:29:31.4.5|
Structure
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