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TargetMu-type opioid receptor
LigandBDBM50336672
Substrate/Competitorn/a
Meas. Tech.ChEMBL_722917
Ki 0.121±n/a nM
Citation Nemoto, TYamamoto, NWatanabe, AFujii, HHasebe, KNakajima, MMochizuki, HNagase, H Synthesis of 6,14-epoxymorphinan derivatives and their pharmacologies. Bioorg Med Chem19:1205-21 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50336672
NameBDBM50336672
Synonyms:CHEMBL1672473 | N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydroxymorphinan-6alpha-yl)methyl]-3-hydroxybenzamide
TypeSmall organic molecule
Emp. Form.C28H32N2O4
Mol. Mass.460.5647
SMILESOc1cccc(c1)C(=O)NC[C@@]12CC[C@@]3(O1)[C@H]1Cc4ccc(O)cc4[C@]3(C2)CCN1CC1CC1 |r,THB:30:29:14:24.18.17|
Structure
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