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Target
Mu-type opioid receptor
Ligand
BDBM50336675
Substrate
n/a
Meas. Tech.
ChEMBL_722917 (CHEMBL1674428)
Ki
4.38±n/a nM
Citation
 Nemoto, T; Yamamoto, N; Watanabe, A; Fujii, H; Hasebe, K; Nakajima, M; Mochizuki, H; Nagase, H Synthesis of 6,14-epoxymorphinan derivatives and their pharmacologies. Bioorg Med Chem 19:1205-21 (2011) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50336675
Synonyms:
CHEMBL1672482 | N-[(17-Benzyl-6beta,14beta-epoxy-3-hydroxymorphinan-6alpha-yl)methyl]benzamide
Type:
Small organic molecule
Emp. Form.:
C31H32N2O3
Mol. Mass.:
480.5974
SMILES:
Oc1ccc2C[C@H]3N(Cc4ccccc4)CC[C@@]4(C[C@]5(CNC(=O)c6ccccc6)CC[C@@]34O5)c2c1 |r,THB:8:7:32:34.4.5|
Structure:
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