Reaction Details Report a problem with these data
Target
HLA class II histocompatibility antigen, DR beta 3 chain
Ligand
BDBM50366439
Substrate
n/a
Meas. Tech.
ChEMBL_47860 (CHEMBL660107)
IC50
178±n/a nM
Citation
Hanson, GJ; Vuletich, JL; Bedell, LJ; Bono, CP; Howard, SC; Welply, JK; Woulfe, SL; Zacheis, ML Design of MHC class II (DR4) ligands using conformationally restricted imino acids at p3 and p5 Bioorg Med Chem Lett 6:1931-1936 (1996) Article
More Info.:
Target
Name:
HLA class II histocompatibility antigen, DR beta 3 chain
Synonyms:
DRB3_HUMAN | HLA class II histocompatibility antigen DRB3-1 | HLA class II histocompatibility antigen, DRB3-1 beta chain | HLA-DRB3 | Human leukocyte antigen DR beta chain | MHC class I antigen DRB3*1
Type:
PROTEIN
Mol. Mass.:
29969.73
Organism:
Homo sapiens (Human)
Description:
ChEMBL_47860
Residue:
266
Sequence:
MVCLKLPGGSSLAALTVTLMVLSSRLAFAGDTRPRFLELRKSECHFFNGTERVRYLDRYFHNQEEFLRFDSDVGEYRAVTELGRPVAESWNSQKDLLEQKRGRVDNYCRHNYGVGESFTVQRRVHPQVTVYPAKTQPLQHHNLLVCSVSGFYPGSIEVRWFRNGQEEKAGVVSTGLIQNGDWTFQTLVMLETVPRSGEVYTCQVEHPSVTSALTVEWRARSESAQSKMLSGVGGFVLGLLFLGAGLFIYFRNQKGHSGLQPTGFLS