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Target
Mu-type opioid receptor
Ligand
BDBM50008854
Substrate
n/a
Meas. Tech.
ChEMBL_146262 (CHEMBL757486)
Ki
410±n/a nM
Citation
 Halfpenny, PR; Horwell, DC; Hughes, J; Humblet, C; Hunter, JC; Neuhaus, D; Rees, DC Highly selective kappa opioid analgesics. 4. Synthesis of some conformationally restricted naphthalene derivatives with high receptor affinity and selectivity. J Med Chem 34:190-4 (1991) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50008854
Synonyms:
2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cyclohexyl)-acetamide; hydrochloride | CHEMBL543331
Type:
Small organic molecule
Emp. Form.:
C21H28N2OS
Mol. Mass.:
356.525
SMILES:
CN([C@H]1CCCC[C@@H]1N1CCCC1)C(=O)Cc1cccc2sccc12
Structure:
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