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Target
Muscarinic acetylcholine receptor M2
Ligand
BDBM50010098
Substrate
n/a
Meas. Tech.
ChEBML_140189
Ki
432±n/a nM
Citation
 Hudkins, RL; DeHaven-Hudkins, DL; Stubbins, JF Muscarinic receptor binding profile of para-substituted caramiphen analogues. J Med Chem 34:2984-9 (1991) [PubMed]  Article 
Target
Name:
Muscarinic acetylcholine receptor M2
Synonyms:
ACM2_RAT | Cholinergic, muscarinic M2 | Chrm-2 | Chrm2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
51555.53
Organism:
RAT
Description:
P10980
Residue:
466
Sequence:
MNNSTNSSNNGLAITSPYKTFEVVFIVLVAGSLSLVTIIGNILVMVSIKVNRHLQTVNNYFLFSLACADLIIGVFSMNLYTLYTVIGYWPLGPVVCDLWLALDYVVSNASVMNLLIISFDRYFCVTKPLTYPVKRTTKMAGMMIAAAWVLSFILWAPAILFWQFIVGVRTVEDGECYIQFFSNAAVTFGTAIAAFYLPVIIMTVLYWHISRASKSRIKKEKKEPVANQDPVSPSLVQGRIVKPNNNNMPGGDGGLEHNKIQNGKAPRDGVTENCVQGEEKESSNDSTSVSAVASNMRDDEITQDENTVSTSLGHSRDDNSKQTCIKIVTKAQKGDVCTPTSTTVELVGSSGQNGDEKQNIVARKIVKMTKQPAKKKPPPSREKKVTRTILAILLAFIITWAPYNVMVLINTFCAPCIPNTVWTIGYWLCYINSTINPACYALCNATFKKTFKHLLMCHYKNIGATR
  
Inhibitor
Name:
BDBM50010098
Synonyms:
1-(4-Tetrazol-1-yl-phenyl)-cyclopentanecarboxylic acid 2-diethylamino-ethyl ester; hydrochloride | CHEMBL542915
Type:
Small organic molecule
Emp. Form.:
C19H27N5O2
Mol. Mass.:
357.45
SMILES:
CCN(CC)CCOC(=O)C1(CCCC1)c1ccc(cc1)-n1cnnn1
Structure:
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