Reaction Details Report a problem with these data
Target
Mu-type opioid receptor
Ligand
BDBM50453050
Substrate
n/a
Meas. Tech.
ChEMBL_147104 (CHEMBL882760)
IC50
12300±n/a nM
Citation
Hruby, VJ; Toth, G; Gehrig, CA; Kao, LF; Knapp, R; Lui, GK; Yamamura, HI; Kramer, TH; Davis, P; Burks, TF Topographically designed analogues of [D-Pen,D-Pen5]enkephalin. J Med Chem 34:1823-30 (1991) [PubMed] Article
More Info.:
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI