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Targetmu/kappa opioid receptor
LigandBDBM50000296
Substrate/Competitorn/a
Meas. Tech.ChEBML_146266
Ki 206±n/a nM
Citation Choi, HMurray, TFDeLander, GECaldwell, VAldrich, JV N-terminal alkylated derivatives of [D-Pro10]dynorphin A-(1-11) are highly selective for kappa-opioid receptors. J Med Chem35:4638-9 (1993) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
mu/kappa opioid receptor
Name:mu/kappa opioid receptor
Synonyms:Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:OPIATE Mu OPRM1 GUINEA PIG::P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50000296
NameBDBM50000296
Synonyms:CHEMBL441765 | CHEMBL482811 | U-50488H
TypeSmall organic molecule
Emp. Form.C19H26Cl2N2O
Mol. Mass.369.329
SMILESCN([C@@H]1CCCC[C@H]1N1CCCC1)C(=O)Cc1ccc(Cl)c(Cl)c1 |r|
Structure
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