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Target
Mu-type opioid receptor
Ligand
BDBM50000651
Substrate
n/a
Meas. Tech.
ChEBML_145295
Ki
3400±n/a nM
Citation
 Heyl, DL; Mosberg, HI Substitution on the Phe3 aromatic ring in cyclic delta opioid receptor-selective dermorphin/deltorphin tetrapeptide analogues: electronic and lipophilic requirements for receptor affinity. J Med Chem 35:1535-41 (1992) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50000651
Synonyms:
10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-(3-hydroxy-benzyl)-3,3-dimethyl-6,9-dioxo-1,2-dithia-5,8-diaza-cycloundecane-4-carboxylic acid | CHEMBL39647
Type:
Small organic molecule
Emp. Form.:
C26H32N4O7S2
Mol. Mass.:
576.685
SMILES:
CC1(C)SSC[C@H](NC(=O)[C@@H](N)Cc2ccc(O)cc2)C(=O)N[C@@H](Cc2cccc(O)c2)C(=O)N[C@@H]1C(O)=O
Structure:
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