Reaction Details Report a problem with these data
Target
Mu-type opioid receptor
Ligand
BDBM82551
Substrate
n/a
Meas. Tech.
ChEMBL_149477 (CHEMBL758227)
Ki
28.4±n/a nM
Citation
Lu, Y; Nguyen, TM; Weltrowska, G; Berezowska, I; Lemieux, C; Chung, NN; Schiller, PW [2',6'-Dimethyltyrosine]dynorphin A(1-11)-NH2 analogues lacking an N-terminal amino group: potent and selective kappa opioid antagonists. J Med Chem 44:3048-53 (2001) [PubMed] Article
More Info.:
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI