Reaction Details Report a problem with these data
Target
Adenylosuccinate synthetase isozyme 2
Ligand
BDBM50149248
Substrate
n/a
Meas. Tech.
ChEMBL_29913 (CHEMBL641276)
IC50
3500±n/a nM
Citation
Erlanson, DA; McDowell, RS; O'Brien, T Fragment-based drug discovery. J Med Chem 47:3463-82 (2004) [PubMed] Article
More Info.:
Target
Name:
Adenylosuccinate synthetase isozyme 2
Synonyms:
ADSS | ADSS2 | AMPSase 2 | AdSS 2 | Adenylosuccinate synthetase 2 | Adenylosuccinate synthetase isozyme 2 | Adenylosuccinate synthetase, acidic isozyme | IMP--aspartate ligase 2 | PURA2_HUMAN
Type:
PROTEIN
Mol. Mass.:
50096.76
Organism:
Homo sapiens (Human)
Description:
ChEMBL_29913
Residue:
456
Sequence:
MAFAETYPAASSLPNGDCGRPRARPGGNRVTVVLGAQWGDEGKGKVVDLLAQDADIVCRCQGGNNAGHTVVVDSVEYDFHLLPSGIINPNVTAFIGNGVVIHLPGLFEEAEKNVQKGKGLEGWEKRLIISDRAHIVFDFHQAADGIQEQQRQEQAGKNLGTTKKGIGPVYSSKAARSGLRMCDLVSDFDGFSERFKVLANQYKSIYPTLEIDIEGELQKLKGYMEKIKPMVRDGVYFLYEALHGPPKKILVEGANAALLDIDFGTYPFVTSSNCTVGGVCTGLGMPPQNVGEVYGVVKAYTTRVGIGAFPTEQDNEIGELLQTRGREFGVTTGRKRRCGWLDLVLLKYAHMINGFTALALTKLDILDMFTEIKVGVAYKLDGEIIPHIPANQEVLNKVEVQYKTLPGWNTDISNARAFKELPVNAQNYVRFIEDELQIPVKWIGVGKSRESMIQLF