Reaction Details Report a problem with these data
Target
Sigma non-opioid intracellular receptor 1
Ligand
BDBM50398057
Substrate
n/a
Meas. Tech.
ChEMBL_873466 (CHEMBL2186561)
Ki
0.960±n/a nM
Citation
James, ML; Shen, B; Zavaleta, CL; Nielsen, CH; Mesangeau, C; Vuppala, PK; Chan, C; Avery, BA; Fishback, JA; Matsumoto, RR; Gambhir, SS; McCurdy, CR; Chin, FT New positron emission tomography (PET) radioligand for imagings-1 receptors in living subjects. J Med Chem 55:8272-82 (2012) [PubMed] Article
More Info.:
Target
Name:
Sigma non-opioid intracellular receptor 1
Synonyms:
Opioid receptor | Oprs1 | SGMR1_RAT | Sigma | Sigma non-opioid intracellular receptor 1 | Sigma opioid receptor | Sigma-1 | Sigmar1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25266.54
Organism:
RAT
Description:
Q9R0C9
Residue:
223
Sequence:
MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSRLIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRYWAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPSTLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP