Reaction Details Report a problem with these data
Target
Cannabinoid receptor 1
Ligand
BDBM50404269
Substrate
n/a
Meas. Tech.
ChEBML_46615
EC50
39811±n/a nM
Citation
 Parkkari, T; Savinainen, JR; Rauhala, AL; Tolonen, TL; Nevalainen, T; Laitinen, JT; Gynther, J; Järvinen, T Synthesis and CB1 receptor activities of novel arachidonyl alcohol derivatives. Bioorg Med Chem Lett 14:3231-4 (2004) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 1
Synonyms:
Brain-type cannabinoid receptor | CANNABINOID CB1 | CB-R | CB1 | CNR1_RAT | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cnr1 | Skr6
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
52856.55
Organism:
Rattus norvegicus (rat)
Description:
P20272
Residue:
473
Sequence:
MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQEKMTAGDNSPLVPAGDTTNITEFYNKSLSSFKENEENIQCGENFMDMECFMILNPSQQLAIAVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHVFHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLMWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIVYAYMYILWKAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLLAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQPLDNSMGDSDCLHKHANNTASMHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
  
Inhibitor
Name:
BDBM50404269
Synonyms:
CHEMBL320549
Type:
Small organic molecule
Emp. Form.:
C23H38O4
Mol. Mass.:
378.5454
SMILES:
CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCCOC(=O)[C@@H](O)CO
Structure:
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