Reaction Details Report a problem with these data
Target
Granzyme K
Ligand
BDBM50187800
Substrate
n/a
Meas. Tech.
ChEMBL_371006 (CHEMBL868504)
Ki
>150000±n/a nM
Citation
Palmer, JT; Rydzewski, RM; Mendonca, RV; Sperandio, D; Spencer, JR; Hirschbein, BL; Lohman, J; Beltman, J; Nguyen, M; Liu, L Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors. Bioorg Med Chem Lett 16:3434-9 (2006) [PubMed] Article
More Info.:
Target
Name:
Granzyme K
Synonyms:
Fragmentin-3 | GRAK_HUMAN | GZMK | Granzyme-3 | NK-TRYP-2 | NK-tryptase-2 | TRYP2
Type:
PROTEIN
Mol. Mass.:
28902.79
Organism:
Homo sapiens (Human)
Description:
ChEMBL_162618
Residue:
264
Sequence:
MTKFSSFSLFFLIVGAYMTHVCFNMEIIGGKEVSPHSRPFMASIQYGGHHVCGGVLIDPQWVLTAAHCQYRFTKGQSPTVVLGAHSLSKNEASKQTLEIKKFIPFSRVTSDPQSNDIMLVKLQTAAKLNKHVKMLHIRSKTSLRSGTKCKVTGWGATDPDSLRPSDTLREVTVTVLSRKLCNSQSYYNGDPFITKDMVCAGDAKGQKDSCKGDSGGPLICKGVFHAIVSGGHECGVATKPGIYTLLTKKYQTWIKSNLVPPHTN