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Target
Acetylcholine-binding protein
Ligand
BDBM50425042
Substrate
n/a
Meas. Tech.
ChEMBL_936605 (CHEMBL2318768)
Ki
79±n/a nM
Citation
 Ussing, CA; Hansen, CP; Petersen, JG; Jensen, AA; Rohde, LA; Ahring, PK; Nielsen, EŘ; Kastrup, JS; Gajhede, M; Frølund, B; Balle, T Synthesis, pharmacology, and biostructural characterization of novela4ß2 nicotinic acetylcholine receptor agonists. J Med Chem 56:940-51 (2013) [PubMed]  Article 
Target
Name:
Acetylcholine-binding protein
Synonyms:
ACHP_LYMST | ACh-binding protein | Acetylcholine Binding protein | Acetylcholine-binding protein (AchBP) | Acetylcholine-binding protein (Ls-AchBP) | AchBP
Type:
n/a
Mol. Mass.:
26055.52
Organism:
Lymnaea stagnalis
Description:
Soluble acetylcholine receptor
Residue:
229
Sequence:
MRRNIFCLACLWIVQACLSLDRADILYNIRQTSRPDVIPTQRDRPVAVSVSLKFINILEVNEITNEVDVVFWQQTTWSDRTLAWNSSHSPDQVSVPISSLWVPDLAAYNAISKPEVLTPQLARVVSDGEVLYMPSIRQRFSCDVSGVDTESGATCRIKIGSWTHHSREISVDPTTENSDDSEYFSQYSRFEILDVTQKKNSVTYSCCPEAYEDVEVSLNFRKKGRSEIL
  
Inhibitor
Name:
BDBM50425042
Synonyms:
(R)-3-(Dimethylamino)Butyl Dimethylcarbamate | CHEMBL2312568
Type:
Small organic molecule
Emp. Form.:
C9H20N2O2
Mol. Mass.:
188.2673
SMILES:
C[C@H](CCOC(=O)N(C)C)N(C)C |r|
Structure:
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