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Target
Delta-type opioid receptor
Ligand
BDBM50189136
Substrate
n/a
Meas. Tech.
ChEMBL_1521809 (CHEMBL3626669)
Ki
>1000±n/a nM
Citation
 Lee, DY; Deng, G; Ma, Z; Xu, W; Yang, L; Liu, J; Dai, R; Liu-Chen, LY Synthesis and biological evaluation of 2-alkyl-2-methoxymethyl-salvinorin ethers as selectiveż-opioid receptor agonists. Bioorg Med Chem Lett 25:4689-92 (2015) [PubMed]  Article 
Target
Name:
Delta-type opioid receptor
Synonyms:
DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40577.25
Organism:
MOUSE
Description:
P32300
Residue:
372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTACTPSDGPGGGAAA
  
Inhibitor
Name:
BDBM50189136
Synonyms:
CHEMBL424698 | Salvinorin B
Type:
Small organic molecule
Emp. Form.:
C21H26O7
Mol. Mass.:
390.4269
SMILES:
COC(=O)[C@@H]1C[C@H](O)C(=O)[C@H]2[C@@]1(C)CC[C@H]1C(=O)O[C@@H](C[C@]21C)c1ccoc1
Structure:
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