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Target
Probable G-protein coupled receptor 34
Ligand
BDBM50177140
Substrate
n/a
Meas. Tech.
ChEMBL_1581710 (CHEMBL3816043)
EC50
36±n/a nM
Citation
 Jung, S; Inoue, A; Nakamura, S; Kishi, T; Uwamizu, A; Sayama, M; Ikubo, M; Otani, Y; Kano, K; Makide, K; Aoki, J; Ohwada, T Conformational Constraint of the Glycerol Moiety of Lysophosphatidylserine Affords Compounds with Receptor Subtype Selectivity. J Med Chem 59:3750-76 (2016) [PubMed]  Article 
Target
Name:
Probable G-protein coupled receptor 34
Synonyms:
G protein-coupled receptor 34 | GPR34_MOUSE | Gpr34 | Probable G-protein coupled receptor 34
Type:
PROTEIN
Mol. Mass.:
43201.40
Organism:
Mus musculus
Description:
ChEMBL_102842
Residue:
375
Sequence:
MTTTSVDSWLCSSHGMHFITNYSDQASQNFSGVPNVTSCPMDEKLLSTVLTTFYSVIFLVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAVADLLLIFCLPFRIMYHINQNKWTLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRRAITTKQSIYVCCIVWTVALAGFLTMIILTLKKGGHNSTMCFHYRDRHNAKGEAIFNFVLVVMFWLIFLLIILSYIKIGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCYWKEIIHKTNEIMLVFSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQSEASRSESTSEFKPGHSLHDLSVTVKMPQYSTKGN
  
Inhibitor
Name:
BDBM50177140
Synonyms:
CHEMBL3814525
Type:
Small organic molecule
Emp. Form.:
C31H35ClNO11P
Mol. Mass.:
664.036
SMILES:
N[C@@H](COP(O)(=O)O[C@@H]1CCCO[C@@H]1COC(=O)CCc1ccccc1OCc1cccc(Oc2ccc(Cl)cc2)c1)C(O)=O |r|
Structure:
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