Reaction Details Report a problem with these data
Target
Leukotriene B4 receptor 1
Ligand
BDBM50213057
Substrate
n/a
Meas. Tech.
ChEMBL_99497 (CHEMBL705027)
Ki
3.0±n/a nM
Citation
  TBA Bioorg Med Chem Lett 4:795-800 (1994)   
Target
Name:
Leukotriene B4 receptor 1
Synonyms:
BLT | BLT1 | BLTR | CMKRL1 | Chemoattractant receptor-like 1 | G-protein coupled receptor 16 | GPR16 | LT4R1_HUMAN | LTB4-R 1 | LTB4R | Leukotriene B4 R1 | Leukotriene B4 receptor | Leukotriene B4 receptor 1 | P2RY7 | P2Y purinoceptor 7 | P2Y7
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37582.68
Organism:
Homo sapiens (Human)
Description:
Q15722
Residue:
352
Sequence:
MNTTSSAAPPSLGVEFISLLAIILLSVALAVGLPGNSFVVWSILKRMQKRSVTALMVLNLALADLAVLLTAPFFLHFLAQGTWSFGLAGCRLCHYVCGVSMYASVLLITAMSLDRSLAVARPFVSQKLRTKAMARRVLAGIWVLSFLLATPVLAYRTVVPWKTNMSLCFPRYPSEGHRAFHLIFEAVTGFLLPFLAVVASYSDIGRRLQARRFRRSRRTGRLVVLIILTFAAFWLPYHVVNLAEAGRALAGQAAGLGLVGKRLSLARNVLIALAFLSSSVNPVLYACAGGGLLRSAGVGFVAKLLEGTGSEASSTRRGGSLGQTARSGPAALEPGPSESLTASSPLKLNELN
  
Inhibitor
Name:
BDBM50213057
Synonyms:
CHEMBL167520
Type:
Small organic molecule
Emp. Form.:
C23H29FN4O2
Mol. Mass.:
412.5004
SMILES:
CCc1cc(c(O)cc1OCCCCCC(C)(C)c1nn[nH]n1)-c1ccc(F)cc1
Structure:
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