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Target
Similar to alpha-tubulin isoform 1
Ligand
BDBM50230728
Substrate
n/a
Meas. Tech.
ChEMBL_211322 (CHEMBL818981)
IC50
26000±n/a nM
Citation
 Terada, T; Fujimoto, K; Nomura, M; Yamashita, J; Wierzba, K; Yamazaki, R; Shibata, J; Sugimoto, Y; Yamada, Y; Kobunai, T Antitumor agents. 3. Synthesis and biological activity of 4 beta-alkyl derivatives containing hydroxy, amino, and amido groups of 4'-O-demethyl-4-desoxypodophyllotoxin as antitumor agents. J Med Chem 36:1689-99 (1993) [PubMed]  Article 
Target
Name:
Similar to alpha-tubulin isoform 1
Synonyms:
Similar to alpha-tubulin isoform 1
Type:
PROTEIN
Mol. Mass.:
10383.05
Organism:
Bos taurus
Description:
ChEMBL_104716
Residue:
99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
  
Inhibitor
Name:
BDBM50230728
Synonyms:
CHEMBL297274
Type:
Small organic molecule
Emp. Form.:
C24H26O8
Mol. Mass.:
442.4584
SMILES:
[H][C@@]12C(COC1=O)[C@H](CCCO)c1cc3OCOc3cc1[C@H]2c1cc(OC)c(O)c(OC)c1
Structure:
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