Target
Neuropeptide Y receptor type 1
Ligand
BDBM82276
Substrate
n/a
Ki
0.54±n/a nM
Comments
PDSP_1380
Citation
 Weinberg, DHSirinathsinghji, DJTan, CPShiao, LLMorin, NRigby, MRHeavens, RHRapoport, DRBayne, MLCascieri, MAStrader, CDLinemeyer, DLMacNeil, DJ Cloning and expression of a novel neuropeptide Y receptor. J Biol Chem 271:16435-8 (1996) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1R_MOUSE | Npy1r
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44024.83
Organism:
MOUSE
Description:
NPY-Y1 NPY1R MOUSE::Q04573
Residue:
382
Sequence:
MNSTLFSKVENHSIHYNASENSPLLAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAVMCLPFTFVYTLMDHWVFGETMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGITVIWVLAVASSLPFVIYQILTDEPFQNVSLAAFKDKYVCFDKFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKIRDSKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKISMNDNEKV
  
Inhibitor
Name:
BDBM82276
Synonyms:
L31,P34-NPY,human | NPY Leu31, Pro34, human, rat | NPY [Leu31, Pro34], human | NPY, LP, porcine | NPY,[Leu31,Pro34] | NPY,[leu31,Pro34], porcine
Type:
Small organic molecule
Emp. Form.:
C188H282N54O56S
Mol. Mass.:
4226.644
SMILES:
n/a
Structure:
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