Target
Neuropeptide Y receptor type 1
Ligand
BDBM82287
Substrate
n/a
Ki
2.1±n/a nM
Comments
PDSP_1387
Citation
 Weinberg, DHSirinathsinghji, DJTan, CPShiao, LLMorin, NRigby, MRHeavens, RHRapoport, DRBayne, MLCascieri, MAStrader, CDLinemeyer, DLMacNeil, DJ Cloning and expression of a novel neuropeptide Y receptor. J Biol Chem 271:16435-8 (1996) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1R_MOUSE | Npy1r
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44024.83
Organism:
MOUSE
Description:
NPY-Y1 NPY1R MOUSE::Q04573
Residue:
382
Sequence:
MNSTLFSKVENHSIHYNASENSPLLAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAVMCLPFTFVYTLMDHWVFGETMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGITVIWVLAVASSLPFVIYQILTDEPFQNVSLAAFKDKYVCFDKFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKIRDSKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKISMNDNEKV
  
Inhibitor
Name:
BDBM82287
Synonyms:
NPY2-36 | NPY2-36, human | NPY2-36, porcine
Type:
Small organic molecule
Emp. Form.:
C181H278N54O55
Mol. Mass.:
4090.4728
SMILES:
n/a
Structure:
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