Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 4
Ligand
BDBM84991
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_1673
Citation
 Baxter, GS Novel discriminatory ligands for 5-HT2B receptors. Behav Brain Res 73:149-52 (1996) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 4
Synonyms:
5-HT4 | 5-hydroxytryptamine receptor 4 | 5HT4R_PIG | HTR4
Type:
Enzyme Catalytic Domain
Mol. Mass.:
15633.90
Organism:
PIGLET
Description:
5-HT4 HTR4 PIGLET::Q29006
Residue:
137
Sequence:
CCQPLVYRNKMTPLRVAVLLAGCWAIPVLISFLPIMQGWNNIGITDLIEKRKFHQNSNSTYCIFMVNKPYAITCSVVAFYIPFLLMVLAYWRIYVTAKEHAHQIQMLQRAGAPAEGRPPSADQHSTHRMRTETKAAK
  
Inhibitor
Name:
BDBM84991
Synonyms:
CAS_3277600 | NSC_3277600 | SB204741
Type:
Small organic molecule
Emp. Form.:
C14H14N4OS
Mol. Mass.:
286.352
SMILES:
Cc1cc(NC(=O)Nc2ccc3n(C)ccc3c2)sn1
Structure:
Search PDB for entries with ligand similarity: