Target
Neuropeptide Y receptor type 5
Ligand
BDBM82276
Substrate
n/a
Ki
0.88±n/a nM
Comments
PDSP_3391
Citation
 Hu, YBloomquist, BTCornfield, LJDeCarr, LBFlores-Riveros, JRFriedman, LJiang, PLewis-Higgins, LSadlowski, YSchaefer, JVelazquez, NMcCaleb, ML Identification of a novel hypothalamic neuropeptide Y receptor associated with feeding behavior. J Biol Chem 271:26315-9 (1996) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 5
Synonyms:
NPY-Y5 | NPY-Y5 receptor | NPY5-R | NPY5R | NPY5R_HUMAN | NPYR5 | NPYY5 | Neuropeptide Y receptor type 5 | Neuropeptide Y receptor type 5 ( NPY Y5) | Y5 receptor
Type:
Enzyme
Mol. Mass.:
50746.64
Organism:
Homo sapiens (Human)
Description:
Q15761
Residue:
445
Sequence:
MDLELDEYYNKTLATENNTAATRNSDFPVWDDYKSSVDDLQYFLIGLYTFVSLLGFMGNLLILMALMKKRNQKTTVNFLIGNLAFSDILVVLFCSPFTLTSVLLDQWMFGKVMCHIMPFLQCVSVLVSTLILISIAIVRYHMIKHPISNNLTANHGYFLIATVWTLGFAICSPLPVFHSLVELQETFGSALLSSRYLCVESWPSDSYRIAFTISLLLVQYILPLVCLTVSHTSVCRSISCGLSNKENRLEENEMINLTLHPSKKSGPQVKLSGSHKWSYSFIKKHRRRYSKKTACVLPAPERPSQENHSRILPENFGSVRSQLSSSSKFIPGVPTCFEIKPEENSDVHELRVKRSVTRIKKRSRSVFYRLTILILVFAVSWMPLHLFHVVTDFNDNLISNRHFKLVYCICHLLGMMSCCLNPILYGFLNNGIKADLVSLIHCLHM
  
Inhibitor
Name:
BDBM82276
Synonyms:
L31,P34-NPY,human | NPY Leu31, Pro34, human, rat | NPY [Leu31, Pro34], human | NPY, LP, porcine | NPY,[Leu31,Pro34] | NPY,[leu31,Pro34], porcine
Type:
Small organic molecule
Emp. Form.:
C188H282N54O56S
Mol. Mass.:
4226.644
SMILES:
n/a
Structure:
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