Reaction Details Report a problem with these data
Target
Melanocortin receptor 4
Ligand
BDBM82410
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_2963
Citation
 Schiöth, HB; Muceniece, R; Wikberg, JE Characterisation of the melanocortin 4 receptor by radioligand binding. Pharmacol Toxicol 79:161-5 (1996) [PubMed]  Article 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM82410
Synonyms:
CAS_50913-82-1 | ORG2766 | Org 2766
Type:
Small organic molecule
Emp. Form.:
C34H51N9O11S
Mol. Mass.:
793.887
SMILES:
CCC(N)C(=O)OC(=O)[C@H](C)N(C(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1ccccc1)C(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](N)CC(C(O)=O)S(C)(=O)=O |r|
Structure:
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