Target
Galanin receptor type 3
Ligand
BDBM85163
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_876
Citation
 Wang, SHe, CHashemi, TBayne, M Cloning and expressional characterization of a novel galanin receptor. Identification of different pharmacophores within galanin for the three galanin receptor subtypes. J Biol Chem 272:31949-52 (1997) [PubMed]  Article 
Target
Name:
Galanin receptor type 3
Synonyms:
GALR3_RAT | Galanin R3 | Galanin receptor type 3 | Galnr3 | Galr3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40439.51
Organism:
RAT
Description:
Galanin R3 GALR3 RAT::O88626
Residue:
370
Sequence:
MADIQNISLDSPGSVGAVAVPVIFALIFLLGMVGNGLVLAVLLQPGPSAWQEPRSTTDLFILNLAVADLCFILCCVPFQAAIYTLDAWLFGAFVCKTVHLLIYLTMYASSFTLAAVSLDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLCFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYSLASRHFRARFRRLWPCGRRRHRHHHRAHRALRRVQPASSGPAGYPGDARPRGWSMEPRGDALRGGGETRLTLSPRGPQ
  
Inhibitor
Name:
BDBM85163
Synonyms:
GMAP (1-41)
Type:
Small organic molecule
Emp. Form.:
C206H327N57O63S
Mol. Mass.:
4642.21
SMILES:
n/a
Structure:
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