Reaction Details
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Report a problem with these dataTarget
Neuropeptide Y receptor type 1
Ligand
BDBM84996
Substrate
n/a
Ki
4.9±n/a nM
Comments
PDSP_2993
Citation
Berglund, MM; Holmberg, SK; Eriksson, H; Gedda, K; Maffrand, JP; Serradeil-Le Gal, C; Chhajlani, V; Grundemar, L; Larhammar, D The cloned guinea pig neuropeptide Y receptor Y1 conforms to other mammalian Y1 receptors. Peptides 20:1043-53 (1999) [PubMed] Article More Info.:
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1R | NPY1R_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44288.14
Organism:
GUINEA PIG
Description:
NPY-Y1 NPY1R GUINEA PIG::Q9WVD0
Residue:
383
Sequence:
MNSTSFSQLENHSVHYNLSEEKPSFFAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLALILIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWIFGEIMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGIAVIWVLAVASSLPFMIYQVLTDEPFQNVTLDAFKDKLVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDSKYRSSESKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPLAFKKISCVENEKI
Inhibitor
Name:
BDBM84996
Synonyms:
BIBP3226 | CAS_5311023 | NSC_5311023
Type:
Small organic molecule
Emp. Form.:
C27H31N5O3
Mol. Mass.:
473.5667
SMILES:
[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6](-[#7]-[#6](=O)-[#6](-c1ccccc1)-c1ccccc1)-[#6](=O)-[#7]-[#6]-c1ccc(-[#8])cc1
Structure:
