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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96907
Substrate
n/a
IC50
28070±n/a nM
Citation
 PubChem, PC Counterscreen for antagonists of the human trace amine associated receptor 1 (hTAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96907
Synonyms:
MLS000332556 | N'-[1-(1H-Indol-3-yl)-meth-(E)-ylidene]-hydrazinecarbodithioic acid methyl ester | N-[[(Z)-3-indolylidenemethyl]amino]carbamodithioic acid methyl ester | N-[[(Z)-indol-3-ylidenemethyl]amino]carbamodithioic acid methyl ester | SMR000221755 | cid_6538175 | methyl N-[[(Z)-indol-3-ylidenemethyl]amino]carbamodithioate
Type:
Small organic molecule
Emp. Form.:
C11H11N3S2
Mol. Mass.:
249.355
SMILES:
CSC(=S)NN=Cc1c[nH]c2ccccc12 |w:5.4|
Structure:
Search PDB for entries with ligand similarity: