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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96655
Substrate
n/a
IC50
9793±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96655
Synonyms:
(6E)-4-chloranyl-6-[(2-phenylethylamino)methylidene]cyclohexa-2,4-dien-1-one | (6E)-4-chloro-6-[(2-phenylethylamino)methylidene]-1-cyclohexa-2,4-dienone | (6E)-4-chloro-6-[(2-phenylethylamino)methylidene]cyclohexa-2,4-dien-1-one | (6E)-4-chloro-6-[(phenethylamino)methylene]cyclohexa-2,4-dien-1-one | 4-chloro-2-{[(2-phenylethyl)imino]methyl}phenol | MLS000699009 | SMR000230665 | cid_6508103
Type:
Small organic molecule
Emp. Form.:
C15H14ClNO
Mol. Mass.:
259.731
SMILES:
Oc1ccc(Cl)cc1C=NCCc1ccccc1 |w:9.10|
Structure:
Search PDB for entries with ligand similarity: