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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96700
Substrate
n/a
IC50
>29875±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96700
Synonyms:
3-chloranyl-5-(2-phenylethylamino)-1,2-thiazole-4-carbonitrile | 3-chloro-5-(2-phenylethylamino)-1,2-thiazole-4-carbonitrile | 3-chloro-5-(2-phenylethylamino)-4-isothiazolecarbonitrile | 3-chloro-5-(phenethylamino)-4-isothiazolecarbonitrile | 3-chloro-5-(phenethylamino)isothiazole-4-carbonitrile | MLS000696339 | SMR000337537 | cid_3787753
Type:
Small organic molecule
Emp. Form.:
C12H10ClN3S
Mol. Mass.:
263.746
SMILES:
Clc1nsc(NCCc2ccccc2)c1C#N
Structure:
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