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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96851
Substrate
n/a
IC50
>29869±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 antagonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96851
Synonyms:
2-amino-5-isopropyl-N-(2-(thiophen-2-yl)ethyl)thiophene-3-carboxamide | 2-amino-5-isopropyl-N-[2-(2-thienyl)ethyl]thiophene-3-carboxamide | 2-amino-5-propan-2-yl-N-(2-thiophen-2-ylethyl)-3-thiophenecarboxamide | 2-amino-5-propan-2-yl-N-(2-thiophen-2-ylethyl)thiophene-3-carboxamide | 2-azanyl-5-propan-2-yl-N-(2-thiophen-2-ylethyl)thiophene-3-carboxamide | MLS003675913 | SMR002356535 | cid_53383658
Type:
Small organic molecule
Emp. Form.:
C14H18N2OS2
Mol. Mass.:
294.436
SMILES:
CC(C)c1cc(C(=O)NCCc2cccs2)c(N)s1
Structure:
Search PDB for entries with ligand similarity: