Reaction Details Report a problem with these data
Target
Lysine-specific demethylase 4C [1-350]
Ligand
BDBM195610
Substrate
n/a
Meas. Tech.
KDM4C Enzymatic Screening Assay
pH
7.5±n/a
IC50
6.2e+2±n/a nM
Comments
extracted
Citation
Vinogradova, M; Gehling, VS; Gustafson, A; Arora, S; Tindell, CA; Wilson, C; Williamson, KE; Guler, GD; Gangurde, P; Manieri, W; Busby, J; Flynn, EM; Lan, F; Kim, HJ; Odate, S; Cochran, AG; Liu, Y; Wongchenko, M; Yang, Y; Cheung, TK; Maile, TM; Lau, T; Costa, M; Hegde, GV; Jackson, E; Pitti, R; Arnott, D; Bailey, C; Bellon, S; Cummings, RT; Albrecht, BK; Harmange, JC; Kiefer, JR; Trojer, P; Classon, M An inhibitor of KDM5 demethylases reduces survival of drug-tolerant cancer cells. Nat Chem Biol 12:531-8 (2016) [PubMed] Article
More Info.:
Target
Name:
Lysine-specific demethylase 4C [1-350]
Synonyms:
GASC1 | JHDM3C | JMJD2C | KDM4C | KDM4C_HUMAN | KIAA0780 | Lysine-specific demethylase 4C (KDM4C)
Type:
Protein
Mol. Mass.:
40626.08
Organism:
Homo sapiens (Human)
Description:
Q9H3R0; His-tagged recombinant KDM4C (1-350) overexpressed in E. coli(DE3)
Residue:
350
Sequence:
MEVAEVESPLNPSCKIMTFRPSMEEFREFNKYLAYMESKGAHRAGLAKVIPPKEWKPRQCYDDIDNLLIPAPIQQMVTGQSGLFTQYNIQKKAMTVKEFRQLANSGKYCTPRYLDYEDLERKYWKNLTFVAPIYGADINGSIYDEGVDEWNIARLNTVLDVVEEECGISIEGVNTPYLYFGMWKTTFAWHTEDMDLYSINYLHFGEPKSWYAIPPEHGKRLERLAQGFFPSSSQGCDAFLRHKMTLISPSVLKKYGIPFDKITQEAGEFMITFPYGYHAGFNHGFNCAESTNFATVRWIDYGKVAKLCTCRKDMVKISMDIFVRKFQPDRYQLWKQGKDIYTIDHTKPTP