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Target
TSC22 domain family protein 3
Ligand
BDBM476590
Substrate
n/a
Meas. Tech.
GILZ gene assays
IC50
24.2±n/a nM
Citation
 Garbaccio, RM; Kern, JC; Mulhearn, JJ; Brandish, PE Phosphonate linkers and their use to facilitate cellular retention of compounds US Patent  US10869929 Publication Date 12/22/2020 
Target
Name:
TSC22 domain family protein 3
Synonyms:
DSIP-immunoreactive peptide | DSIPI | Delta sleep-inducing peptide immunoreactor | GILZ | Glucocorticoid-induced leucine zipper protein | Protein DIP | T22D3_HUMAN | TSC-22-like protein | TSC-22-related protein | TSC-22R | TSC22D3 | hDIP
Type:
Protein
Mol. Mass.:
14799.51
Organism:
Human
Description:
Q99576
Residue:
134
Sequence:
MNTEMYQTPMEVAVYQLHNFSISFFSSLLGGDVVSVKLDNSASGASVVAIDNKIEQAMDLVKNHLMYAVREEVEILKEQIRELVEKNSQLERENTLLKTLASPEQLEKFQSCLSPEEPAPESPQVPEAPGGSAV
  
Inhibitor
Name:
BDBM476590
Synonyms:
US10869929, Compound 29 | US11554172, Compound 29
Type:
Small organic molecule
Emp. Form.:
C41H59N2O9P
Mol. Mass.:
754.8889
SMILES:
CCCC1O[C@@H]2C[C@H]3[C@@H]4CCC5=Cc6c(C[C@]5(C)[C@H]4[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO)cnn6-c1cccc(OCCCCCCCCCP(O)(O)=O)c1 |r,w:3.2,t:11|
Structure:
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