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Target
Somatostatin receptor type 4
Ligand
BDBM506555
Substrate
n/a
Meas. Tech.
SSTR4 I-125 Somatostatin Competition Binding Assay
IC50
63.1±n/a nM
Citation
 Cheruvallath, Z; Green, J; Johnson, B; Schleicher, K; Sun, H; Tang, M Piperidinyl-3-(aryloxy)propanamides and propanoates US Patent  US11045457 Publication Date 6/29/2021 
Target
Name:
Somatostatin receptor type 4
Synonyms:
SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4)
Type:
Enzyme
Mol. Mass.:
42015.38
Organism:
Homo sapiens (Human)
Description:
P31391
Residue:
388
Sequence:
MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLPIAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRAVALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCMCPPLPCQQEALQPEPGRKRIPLTRTTTF
  
Inhibitor
Name:
BDBM506555
Synonyms:
US11045457, Example 155
Type:
Small organic molecule
Emp. Form.:
C24H30F3N3O2
Mol. Mass.:
449.5091
SMILES:
CN([C@@H]1CCNC[C@H]1c1ccccc1C)C(=O)C(C)(C)COc1ncccc1C(F)(F)F |r|
Structure:
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