Assay Method Information

Assay Name:  Scintillation Proximity Assay (SPA)
Description:  The compound inhibitory activity was determined by incubation with purified PLK enzyme and biotinylated peptide substrate in the presence ATP/[gamma-33P]ATP. After incubation, the phosphorylated substrate was separated from nonincorporated radioactive ATP using SPA beads. Incorporated radioactivity was measured using Packard TopCount.
Affinity data for this assay
 

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