Assay Method Information

Assay Name:  ChEMBL_1645467 (CHEMBL3994396)
Description:  Antagonist activity at human adenosine A1 receptor expressed in HEK293 cells assessed as reduction in CPA-mediated inhibition of forskolin-stimulated cAMP level preincubated for 15 mins followed by CPA treatment for 15 mins and subsequent addition of forskolin measured after 30 mins by HTRF assay
Affinity data for this assay
 

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