Assay Method Information

Assay Name:  ChEMBL_1660309 (CHEMBL4009921)
Description:  Uncompetitive inhibition of human N-terminal His6-SUMO-tagged SIRT2 catalytic domain (43 to 356 residues) deacetylase activity expressed in Escherichia coli using alpha-tubulin-acetylLys40 peptide as substrate up to 5 uM after 45 mins by Lineweaver-Burk double reciprocal plot analysis
Affinity data for this assay
 

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