Assay Method Information | |
| ChEMBL_1621714 (CHEMBL3863997) |
Description: | Antagonist activity at DRD2 (unknown origin) expressed in HEK293T cells transfected with Galphai1-RLuc8 and gamma2-GFP10 assessed as inhibition of quinpirole-induced Gi1 activation pre-incubated with quinpirole for 10 mins before compound incubation for 10 mins by BRET assay |
Affinity data for this assay | |
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