Assay Method Information

Assay Name:  ChEMBL_1621714 (CHEMBL3863997)
Description:  Antagonist activity at DRD2 (unknown origin) expressed in HEK293T cells transfected with Galphai1-RLuc8 and gamma2-GFP10 assessed as inhibition of quinpirole-induced Gi1 activation pre-incubated with quinpirole for 10 mins before compound incubation for 10 mins by BRET assay
Affinity data for this assay
 

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