Assay Method Information

Assay Name:  ChEMBL_1991443 (CHEMBL4625178)
Description:  Binding affinity to murine DNMT3A catalytic domain assessed as enzyme-DNA complex formation at 5 uM using 30-mer duplex DNA (22 AT bp) as substrate preincubated for 30 mins followed by enzyme addition by fluorescence polarization assay (Rvb = 0.4 +/- 0.1 uM)
Affinity data for this assay
 

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