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Targets Binding with 3027 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Disintegrin and metalloproteinase domain-containing protein 17 (ADAM-17)
Ki:
425
IC50:
3215
EC50:
10
128
4
2D
3D
TSV
EDG6
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
Endothelial differentiation G-protein coupled receptor 6
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
Low-voltage-activated calcium channel alpha1 3.2 subunit
Ki:
4
IC50:
1007
Kd:
1
EC50:
786
37
10
2D
3D
TSV
S1P receptor 4
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
S1P receptor Edg-6
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
S1P4
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
Sphingosine 1-phosphate receptor 4
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
Sphingosine 1-phosphate receptor Edg-6
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
sphingosine-1-phosphate 4 S1P4
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
Sphingosine-1-phosphate receptor 4
Ki:
13
IC50:
428
EC50:
334
61
3
2D
3D
TSV
TNF-alpha converting enzyme (TACE)
Ki:
425
IC50:
3215
EC50:
10
128
4
2D
3D
TSV
TNF-alpha-converting enzyme (TACE)
Ki:
425
IC50:
3215
EC50:
10
128
4
2D
3D
TSV
Tumor Necrosis Factor Alpha Converting Enzyme
Ki:
425
IC50:
3215
EC50:
10
128
4
2D
3D
TSV
Tumor necrosis factor-α converting enzyme (TACE)
Ki:
425
IC50:
3215
EC50:
10
128
4
2D
3D
TSV
voltage-dependent T-type calcium channel subunit alpha-1H isoform a
Ki:
4
IC50:
1007
Kd:
1
EC50:
786
37
10
2D
3D
TSV